A-836339, [3H]-

Catalog>7TM>Cannabinoid>[3H]-A-836339

*EXCLUSIVE*

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Product Number: NML3H1023
Alternate Name: NA
Specific Activity: 75-87 Ci/mmol
2.7-3.2TBq/mmol
CAS Number (Parent): 959746-77-1
Shipping Conditions: Shipped on dry ice
Storage Conditions: -20ºC, in ethanol

Information:
Selective Cannabinoid CB2 receptor agonist radioligand.

Reference:
Synthesis and biodistribution of [11C]A-836339, a new potential radioligand for PET imaging of cannabinoid type 2 receptors (CB2).
Horti AG, Gao Y, Ravert HT, Finley P, Valentine H, Wong DF, Endres CJ, Savonenko AV, Dannals RF. (2010) Bioorganic and Medicinal Chemistry 18(14):5202-7. PMID: 20554448

Characterization of a cannabinoid CB2 receptor-selective agonist, A-836339 [2,2,3,3-tetramethyl-cyclopropanecarboxylic acid [3-(2-methoxy-ethyl)-4,5-dimethyl-3H-thiazol-(2Z)-ylidene]-amide], using in vitro pharmacological assays, in vivo pain models, and pharmacological magnetic resonance imaging.
Yao BB, Hsieh G, Daza AV, Fan Y et. al. (2009) Journal of Pharmacology and Experimental Therapeutics 328 (1): 141-151. PMID: 18931146

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