Almorexant, [Methoxy-3H]-

Catalog>7TM>Peptide>OX>[3H]Almorexant

*EXCLUSIVE*

Product Number: NML3H1010
Alternate Name: ACT-078573
Specific Activity: 46-54 Ci/mmol
1.7-2.0 TBq/mmol
CAS Number (Parent): 871224-64-5
Shipping Conditions: Shipped on dry ice
Storage Conditions: -20ºC, in ethanol

Information: Non-selective OX1 & OX2 receptor antagonist radioligand.

Reference:
Mapping the binding pocket of dual antagonist almorexant to human orexin 1 and orexin 2 receptors: Comparison with the selective OX1 antagonist SB-674042 and the selective OX2 antagonist N-ethyl-2-[(6-methoxy-pyridin-3-yl)-(toluene-2- sulfonyl)-amino]-N-pyridin-3-ylmethyl-acetamide (EMPA).
P. Malherbe, O. Roche, A. Marcuz, C. Kratzeisen, J. G. Wettstein, and C. Bissantz. (2010) Molecular Pharmacology 78:81–93. PMID: 20404073

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